GHK-Cu Reference

Copper tripeptide · Research compound (cosmetic use of topical forms)

ClassCopper tripeptide
StatusResearch compound (cosmetic use of topical forms)
Typical vials50 mg, 100 mg
Dose range1 mg to 3 mg
FrequencyDaily
Half-lifeNo human data
Dosing unitmilligrams
RouteSubcutaneous injection

What GHK-Cu is

GHK-Cu is a naturally occurring copper-binding tripeptide with a large literature on skin repair and collagen synthesis, almost all of it topical or in vitro. Injectable use in skin and recovery protocols is a community extrapolation from that work, not something the literature directly supports.

It is the outlier on this page for vial sizes: 50 and 100 mg vials are normal because daily milligram doses burn through a vial quickly. It also stings; the copper complex is acidic relative to most peptides, and slow injection is the usual advice.

What we do not know

  • The human evidence is topical and cosmetic. Injected use, which is what the reconstitution math on this page is for, has no published human trials.
  • Systemic copper load from repeated injection is not characterized.
  • Claimed systemic effects such as organ repair rest on in vitro gene-expression work, not outcomes.

Reconstitution math

Concentration is everything: the same 50 mg vial gives a different draw for every amount of bacteriostatic water you add. The table uses the common 5 mL setup for each vial size, which puts every unit on a U-100 insulin syringe at 100 mcg for the default vial. Dashes mark draws too small to measure or larger than the syringe.

VialBAC waterConcentration1 mg2 mg3 mg
50 mg5 mL10 mg/mL10 u20 u30 u
100 mg5 mL20 mg/mL5 u10 u15 u
GHK-Cu syringe drawsDRAW GUIDEEach dose as a filled syringe50 mg vial + 5 mL bacteriostatic water = 1 mg per 0.1 mL (10 units).0481216202428323640units on a U-100 insulin syringe (first 40 units shown)1 mg10 u (0.1 mL)2 mg20 u (0.2 mL)3 mg30 u (0.3 mL)peprecon.com
Draw positions for the common doses at the default setup.

Dosing and protocol

Community protocol: about 1 to 2 mg daily subcutaneously; sold in much larger vials than other peptides.

Community dosing runs about 1 to 2 mg daily. With a 50 mg vial and 5 mL of bacteriostatic water, 1 mg is 10 units on an insulin syringe. GHK-Cu is a core component of the GLOW and KLOW blends; use the blend calculator when it shares a vial with BPC-157 and TB-500.

Pharmacokinetics

No curve is shown, on purpose.

There is no human pharmacokinetic characterization of injected GHK-Cu. Published human work is largely topical and cosmetic; injection dosing is entirely community convention, so no curve is shown.

How it is thought to work

A copper-binding tripeptide present naturally in plasma, where its concentration falls with age. The copper complex is the active form; it influences collagen synthesis and wound-healing signaling, and is a long-established cosmetic ingredient.

How GHK-Cu is thought to workMECHANISMGHK-Cu: the proposed chainA proposed pathway. The last step is the one that needs evidence in people.1Applied topically, or injected2A copper-binding tripeptide, where the copper complex is the active formPresent naturally in plasma, at concentrations that fall with age.3Collagen synthesis and wound-healing signaling4Skin appearance and wound repairLong established as a cosmetic ingredient, which is a different evidence barfrom a drug.STRONGEST PUBLISHED EVIDENCE FOR ANY CLAIMED OUTCOMEHuman RCTOutcome by outcome, see the table below.peprecon.com

What the evidence supports

This table grades how well each outcome has been studied in humans, not how well GHK-Cu works. A strong grade means the question was asked properly, and the answer may still have been negative. Nothing here is inherited from a drug class, a close analog, or the parent molecule of a fragment.

OutcomeStrongest published evidence
Skin appearance, topicalHuman RCT
Wound healing, topicalHuman, observational
Gene expression changesMechanistic only
Any outcome from injectionNo data
Human RCTAt least one randomized controlled trial in people reports this outcome. The result may still have been negative.
Human, observationalReported in people without randomization: open-label, single-arm, retrospective, or case series.
Mechanistic onlySupported only by cell, tissue or biochemical work, or by reasoning from a related molecule.
No dataNo published evidence at any level that we could find.

Storage and handling

Lyophilized vials keep best cold, dark, and dry; refrigeration is the community default and freezing lyophilized powder is common for long holds. After reconstitution, refrigerate at 2 to 8 C, do not freeze the solution, and date the vial. Bacteriostatic water's preservative keeps multi-dose use practical for about 28 days by USP convention, though our 120-day stability study found the preservative itself outlasts that window.

Reconstituted GHK-Cu is unusually stable by reputation (the copper complex is robust), but the same refrigeration rule applies. The solution is distinctly blue; a color change is a red flag.

Got a certificate of analysis with your vial? Run it through our COA Reader: it reads the report in plain English, checks purity and mass against the label claim, and links the testing lab’s own verification page. Our guide to reading a COA explains what the numbers do and do not tell you.

Sources

  1. Pickart and Margolina, GHK-Cu regenerative and protective actions, Int J Mol Sci 2018
  2. Pickart et al., GHK peptide as a natural modulator of multiple cellular pathways, BioMed Res Int 2015PMID 26236730 · DOI

Related references: BPC-157 · TB-500